Medicamentul anticancer bexaroten a făcut nu doar să dispară la acei şoareci 75% din totalul plăcilor betaamiloide, o formă de proteină a cărei acumulare reprezintă una dintre caracteristicile patologice principale ale maladiei Alzheimer, ci a inversat şi simptome ale bolii, precum pierderile de memorie.
La doar 72 de ore după ce au început tratamentul cu bexaroten, şoarecii de laborator – modificaţi genetic pentru a dezvolta un echivalent al maladiei Alzheimer umane – au început să prezinte comportamente normale, au explicat autorii acestui studiu, publicat în revista Science, citată de Mediafax.
Animalele şi-au regăsit memoria şi simţul mirosului, a explicat medicul Daniel Wesson, profesor adjunct de ştiinţe neuronale la Facultatea de medicină Case Western din Cleveland (Ohio, SUA), principalul autor al studiului.
Această descoperire este „fără precedent”, afirmă Paige Cramer, cercetător la aceeaşi universitate şi colaborator la acest studiu. „Până acum, cel mai bun dintre tratamentele existente pentru şoarecii de laborator avea nevoie de mai multe luni pentru a elimina plăcile amiloide”, a mai spus acesta.
Maladia Alzheimer apare, în majoritatea cazurilor, atunci când organismul, îmbătrânind, îşi pierde capacitatea de a elimina plăcile betaamiloide care se formează în mod natural în creier.
Laboratorul japonez Eisai a cumpărat drepturile de distribuţie pe plan mondial pentru bexaroten, în 2006.
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